Do All Roads Really Lead to Rome? Learnings from Comparative Analysis using SPR, NMR, & X-Ray Crystallography to Optimize Fragment Screening in Drug Discovery.

There are several biophysical methods developed to rapidly identify weakly binding fragments to a target protein. X-ray crystallography provides structural information that is crucial for fragment optimization, however there are several criteria that must be met for a successful fragment screening...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
मुख्य लेखक: Hassaan, Engi
अन्य लेखक: Klebe, Gerhard (Prof. Dr.) (शोध सलाहकार)
स्वरूप: Dissertation
भाषा:अंग्रेज़ी
प्रकाशित: Philipps-Universität Marburg 2019
विषय:
ऑनलाइन पहुंच:पीडीएफ पूर्ण पाठ
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