Ngā hua rapu - Klebe, Gerhard
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Crystallographic Fragment Screening on the Shigella Type III Secretion System Chaperone IpgC mā Gárdonyi, Marina, Hasewinkel, Christian, Wallbaum, Johanna, Wollenhapt, Jan, Weiss, Manfred S., Klebe, Gerhard, Reuter, Klaus, Heine, Andreas
I whakaputaina 2023Kei te kohinga: Publikationen im Open Access gefördert durch die UBTau karanga: es/2024/0803Kuputuhi katoa PDF
Tuhinga -
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Leitstruktursuche mithilfe eines kristallographischen Fragment-Screenings zur Inhibierung des Klasse-II-Chaperons IpgC aus Shigella flexneri mā Gárdonyi, Marina
I whakaputaina 2021Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2021/0513Kuputuhi katoa PDF
Dissertation -
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Optimization of the Drug Design Process by Ligand Preorganization and Occupancy of Transient Binding Pockets Based on the Model Proteins Thrombin and Aldose Reductase mā Sandner, Anna Sophie
I whakaputaina 2022Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2022/0118Kuputuhi katoa PDF
Dissertation -
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Mutational Studies on 17β-HSD14, Serial Synchrotron X-ray Crystallography, Solubility Enhancement using Cyclodextrins and Fragment-Based Drug Discovery Multiple Blocks to Pave the... mā Badran, Mohammed
I whakaputaina 2021Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2021/0095Kuputuhi katoa PDF
Dissertation -
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Neue Ansätze zur Entwicklung von Modulatoren der homodimeren tRNA-Guanin-Transglycosylase mā Nguyen, Andreas
I whakaputaina 2020Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2020/0517Kuputuhi katoa PDF
Dissertation -
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Fragment-basierte Leitstruktursuche am Beispiel der Proteinkinase A mā Oebbeke, Matthias
I whakaputaina 2021Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2021/0112Kuputuhi katoa PDF
Dissertation -
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From Serendipity to the Rational Design of Protein–Protein Interface Modulators Targeting a tRNA-Modifying Enzyme mā Nguyen, Dzung
I whakaputaina 2020Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2021/0067Kuputuhi katoa PDF
Dissertation -
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Thermodynamic, Kinetic and Crystallographic Investigations of Benzenesulfonamides as Ligands of Human Carbonic Anhydrase II mā Glöckner, Steffen
I whakaputaina 2020Ētahi atu kaituhi: “… Klebe, Gerhard Prof. Dr. …”
Tau karanga: diss/z2020/0123Kuputuhi katoa PDF
Dissertation -
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Do All Roads Really Lead to Rome? Learnings from Comparative Analysis using SPR, NMR, & X-Ray Crystallography to Optimize Fragment Screening in Drug Discovery. mā Hassaan, Engi
I whakaputaina 2019Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2019/0491Kuputuhi katoa PDF
Dissertation -
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Synthese von D-Phe/D-DiPhe-Pro-basierenden Liganden und deren biophysikalischen Charakterisierung zur Selektivitätsstudie von Thrombin und Trypsin sowie ein synthetischer Beitrag z... mā Ngo, Trong Khang
I whakaputaina 2020Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2020/0081Kuputuhi katoa PDF
Dissertation -
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Targeting farnesyl pyrophosphate synthase of Trypanosoma cruzi by fragment-based lead discovery mā Petrick, Joy Kristin
I whakaputaina 2019Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2019/0501Kuputuhi katoa PDF
Dissertation -
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Targeting Trypanosoma brucei FPPS by Fragment-based drug discovery mā Münzker Lena
I whakaputaina 2019Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2019/0500Kuputuhi katoa PDF
Dissertation -
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The Power of Fragments: FBLD approach to investigate protein structures mā Magari, Francesca
I whakaputaina 2020Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2020/0214Kuputuhi katoa PDF
Dissertation -
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Identifizierung, Charakterisierung und Untersuchungen der Struktur-Wirkungs-Beziehung sowie des Mode of Action eines neuen antimikrobiellen Peptids aus Hirudo verbana mā Müller, Daniela
I whakaputaina 2019Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr. rer. nat.) …”
Tau karanga: diss/z2019/0250Kuputuhi katoa PDF
Dissertation -
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Expanding the Toolbox for Computational Analysis in Rational Drug Discovery: Using Biomolecular Solvation to Predict Thermodynamic, Kinetic and Structural Properties of Protein-Lig... mā Hüfner, Tobias
I whakaputaina 2019Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2019/0494Kuputuhi katoa PDF
Dissertation -
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Inhibitor Synthesis and Biophysical Characterization of Protein–Ligand–Solvent Interactions An Analysis of the Thermodynamics and Kinetics of Ligand Binding to Thermolysin mā Cramer, Jonathan
I whakaputaina 2017Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2017/0465Kuputuhi katoa PDF
Dissertation -
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Characterisation and differentiation of kinase binding pockets in PKA and PIM1 by small molecule fragments using protein crystallography mā Siefker, Christof
I whakaputaina 2018Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2018/0229Kuputuhi katoa PDF
Dissertation -
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Structural Characterization of 17β-Hydroxysteroid Dehydrogenase Type 14 and Inhibitor Optimization Using Crystallography and Computational Techniques mā Bertoletti, Nicole
I whakaputaina 2017Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2017/0671Kuputuhi katoa PDF
Dissertation -
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Beyond Affinity: Drug-Kinase Interaction Put under the Microscope mā Wienen-Schmidt, Barbara
I whakaputaina 2017Ētahi atu kaituhi: “… Klebe, Gerhard (Prof.) …”
Tau karanga: diss/z2017/0537Kuputuhi katoa PDF
Dissertation -
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Proteindynamik - Flexibilität in Zielproteinen des strukturbasierten Wirkstoffdesigns mā Terwesten, Felix
I whakaputaina 2017Ētahi atu kaituhi: “… Klebe, Gerhard (Prof. Dr.) …”
Tau karanga: diss/z2018/0049Kuputuhi katoa PDF
Dissertation